ubrogepant 100 MG Oral Tablet
Managing this medication for someone you care for? Eleplan keeps diagnoses, medications and appointments in one plan.
Start free with EleplanClinical drug
ubrogepant 100 MG Oral Tablet
100 MG · Oral Tablet · oral
A form of ubrogepant →
ubrogepant 100 MG Oral Tablet — Calcitonin gene-related peptide (CGRP) antagonists. Strength, form, class, interactions & more.

Active ingredient
Classification
Calcitonin gene-related peptide (CGRP) antagonistsCalcitonin Gene-related Peptide Receptor Antagonist
Drug interactions
Ubrogepant has several drug interactions primarily involving CYP3A4 inhibitors and inducers, as well as BCRP and P-gp inhibitors.
- majorstrong CYP3A4 inducers (e.g., phenytoin, barbiturates, rifampin, St. John’s Wort) — loss of ubrogepant efficacy is expected
- majorstrong CYP3A4 inhibitors (e.g., ketoconazole, itraconazole, clarithromycin) — significant increase in exposure of ubrogepant
- moderatemoderate CYP3A4 inhibitors (e.g., cyclosporine, ciprofloxacin, fluconazole, fluvoxamine, grapefruit juice) — increase in ubrogepant exposure
- moderateBCRP and/or P-gp only inhibitors (e.g., quinidine, carvedilol, eltrombopag, curcumin) — may increase the exposure of ubrogepant
Source: RxNorm + openFDA + RxClass + FAERS · 2026
Look up another medication