resmetirom 100 MG Oral Tablet [Rezdiffra]
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resmetirom 100 MG Oral Tablet [Rezdiffra]
100 MG · Oral Tablet · oral
A form of resmetirom →
resmetirom 100 MG Oral Tablet [Rezdiffra] — Liver therapy. Strength, form, class, interactions & more.
![resmetirom 100 MG Oral Tablet [Rezdiffra]](https://dailymed.nlm.nih.gov/dailymed/image.cfm?setid=e67ea09f-a840-439c-86c8-f98585f978b2&name=madrigal-01.jpg)
Active ingredient
Classification
Liver therapyThyroid Hormone Receptor beta Agonist
Drug interactions
Resmetirom has several clinically significant drug interactions, particularly with CYP2C8 inhibitors and substrates, as well as with certain statins.
- majorstrong CYP2C8 inhibitors (e.g., gemfibrozil) — increased risk of adverse reactions
- moderatemoderate CYP2C8 inhibitors (e.g., clopidogrel) — increased risk of adverse reactions
- moderateatorvastatin, pravastatin, rosuvastatin, simvastatin — increased risk of adverse reactions related to statins
- moderateCYP2C8 substrates — increased risk of adverse reactions
Source: RxNorm + openFDA + RxClass + FAERS · 2026
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