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idelalisib 100 MG Oral Tablet [Zydelig]
100 MG · Oral Tablet · oral
A form of idelalisib →
idelalisib 100 MG Oral Tablet [Zydelig] — Phosphatidylinositol-3-kinase (Pi3K) inhibitors. Strength, form, class, interactions & more.
![idelalisib 100 MG Oral Tablet [Zydelig]](https://dailymed.nlm.nih.gov/dailymed/image.cfm?setid=efbdafa9-d18c-4e85-b4a2-1e620fc74e50&name=zydelig-01.jpg)
Active ingredient
Classification
Drug interactions
Idelalisib has significant interactions with strong CYP3A modulators that can affect its concentrations and efficacy.
- majorstrong CYP3A inhibitors — may increase idelalisib concentrations
- majorstrong CYP3A inducers — may decrease idelalisib concentrations
- majorsensitive CYP3A substrates — may increase concentrations of CYP3A substrates
Real-world adverse events (FAERS)
Source: RxNorm + openFDA + RxClass + FAERS · 2026
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