idelalisib 100 MG Oral Tablet
Managing this medication for someone you care for? Eleplan keeps diagnoses, medications and appointments in one plan.
Start free with EleplanClinical drug
idelalisib 100 MG Oral Tablet
100 MG · Oral Tablet · oral
A form of idelalisib →
idelalisib 100 MG Oral Tablet — Phosphatidylinositol-3-kinase (Pi3K) inhibitors. Strength, form, class, interactions & more.

Active ingredient
Classification
Phosphatidylinositol-3-kinase (Pi3K) inhibitorsKinase Inhibitor
Drug interactions
Idelalisib has significant interactions with strong CYP3A modulators that can affect its concentrations and efficacy.
- majorstrong CYP3A inhibitors — may increase idelalisib concentrations
- majorstrong CYP3A inducers — may decrease idelalisib concentrations
- majorsensitive CYP3A substrates — may increase concentrations of CYP3A substrates
Real-world adverse events (FAERS)
Disease Progression1,225Death802Diarrhoea771Off Label Use572Pneumonia437Pyrexia375Drug Ineffective317Fatigue301
Source: RxNorm + openFDA + RxClass + FAERS · 2026
Look up another medication