entrectinib 100 MG Oral Capsule
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entrectinib 100 MG Oral Capsule
100 MG · Oral Capsule · oral
A form of entrectinib →
entrectinib 100 MG Oral Capsule — Other protein kinase inhibitors. Strength, form, class, interactions & more.

Active ingredient
Classification
Other protein kinase inhibitors
Drug interactions
Entrectinib has several drug interactions that require caution or avoidance during coadministration.
- majormoderate or strong CYP3A inhibitors — increases entrectinib plasma concentrations, which could increase the frequency or severity of adverse reactions
- majorgrapefruit products — inhibits CYP3A, potentially increasing entrectinib plasma concentrations
- majormoderate or strong CYP3A inducers — decreases entrectinib plasma concentrations, which may reduce ROZLYTREK efficacy
- majorother products that prolong QT/QTc interval — QTc interval prolongation can occur
Source: RxNorm + openFDA + RxClass + FAERS · 2026
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