apalutamide 240 MG Oral Tablet [Erleada]
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apalutamide 240 MG Oral Tablet [Erleada]
240 MG · Oral Tablet · oral
A form of apalutamide →
apalutamide 240 MG Oral Tablet [Erleada] — Anti-androgens. Strength, form, class, interactions & more.
![apalutamide 240 MG Oral Tablet [Erleada]](https://dailymed.nlm.nih.gov/dailymed/image.cfm?setid=d1cda4f7-cb33-46ea-b9ac-431f6452b1a5&name=Erleada_240+mg_Label.jpg)
Active ingredient
Classification
Anti-androgens
Drug interactions
Apalutamide may interact with various drugs that are substrates of certain enzymes and transporters, potentially affecting their effectiveness.
- unknownCYP3A4 substrates — may result in loss of activity of these medications
- unknownCYP2C19 substrates — may result in loss of activity of these medications
- unknownCYP2C9 substrates — may result in loss of activity of these medications
- unknownP-gp substrates — may result in loss of activity of these medications
- unknownBCRP substrates — may result in loss of activity of these medications
- unknownOATP1B1 substrates — may result in loss of activity of these medications
- moderatestrong CYP2C8 inhibitors — predicted to increase the steady-state exposure of the active moieties
- moderatestrong CYP3A4 inhibitors — predicted to increase the steady-state exposure of the active moieties
Real-world adverse events (FAERS)
Rash1,229Death1,165Fatigue1,130Hot Flush846Product Dose Omission Issue436Asthenia420Diarrhoea391Dizziness359
Source: RxNorm + openFDA + RxClass + FAERS · 2026
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